Data wydania | Tytuł | Autor |
2019 | Bioactivity of Methoxylated and Methylated 1-Hydroxynaphthalene-2-Carboxanilides: Comparative Molecular Surface Analysis | Michnová, Hana; Pospíšilová, Šárka; Gonec, Tomáš; Kapustíková, Iva; Kollár, Peter; Kozik, Violetta; Musioł, Robert; Jendrzejewska, Izabela; Vanco, Jan; Trávnícek, Zdenek; Cížek, Alois; Bąk, Andrzej; Jampílek, Josef |
2020 | Biological activities and ADMET-related properties of novel set of cinnamanilides | Kos, Jiri; Bąk, Andrzej; Kozik, Violetta; Jankech, Timotiej; Strharsky, Tomas; Świetlicka, Aleksandra; Michnova, Hana; Hosek, Jana; Smoliński, Adam; Oravec, Michal; Devinsky, Ferdinand; Hutta, Milan; Jampilek, Josef |
2020 | Biological Evaluation of 3-Benzylidenechromanones and Their Spiropyrazolines-Based Analogues | Adamus-Grabicka, Angelika A.; Markowicz-Piasecka, Magdalena; Cieślak, Marcin; Królewska-Golińska, Karolina; Hikisz, Paweł; Kusz, Joachim; Małecka, Magdalena; Budzisz, Elżbieta |
2021 | Chromatographic and computational screening of lipophilicity and pharmacokinetics of newly synthesized betulin-1,4-quinone hybrids | Kadela-Tomanek, Monika; Jastrzębska, Maria; Chrobak, Elwira; Bębenek, Ewa; Boryczka, Stanisław |
2020 | Consensus-based pharmacophore mapping for new set of N-(disubstitutedphenyl)- 3-hydroxyl-naphthalene-2-carboxamides | Bąk, Andrzej; Kos, Jiri; Michnova, Hana; Gonec, Tomas; Pospisilova, Sarka; Kozik, Violetta; Cizek, Alois; Smoliński, Adam; Jampilek, Josef |
2021 | Lipophilicity, pharmacokinetic properties, and molecular docking study on SARS-CoV-2 target for betulin triazole derivatives with attached 1,4- quinone | Kadela-Tomanek, Monika; Jastrzębska, Maria; Marciniec, Krzysztof; Chrobak, Elwira; Bębenek, Ewa; Boryczka, Stanisław |
2021 | Synthesis and hybrid SAR property modeling of novel cholinesterase inhibitors | Kos, Jiri; Kozik, Violetta; Pindajkova, Dominika; Jankech, Timotiej; Smoliński, Adam; Stepankova, Sarka; Hosek, Jan; Oravec, Michal; Jampilek, Josef; Bąk, Andrzej |
2021 | Towards property profiling: SYNTHESIS and SAR probing of new tetracyclic diazaphenothiazine analogues | Empel, Anna; Bąk, Andrzej; Kozik, Violetta; Latocha, Małgorzata; Cizek, Alois; Jampilek, Josef; Suwińska, Kinga; Sochanik, Aleksander; Zięba, Andrzej |