Issue Date | Title | Author(s) |
2021 | Chromatographic and computational screening of lipophilicity and pharmacokinetics of newly synthesized betulin-1,4-quinone hybrids | Kadela-Tomanek, Monika; Jastrzębska, Maria; Chrobak, Elwira; Bębenek, Ewa; Boryczka, Stanisław |
2021 | Lipophilicity, pharmacokinetic properties, and molecular docking study on SARS-CoV-2 target for betulin triazole derivatives with attached 1,4- quinone | Kadela-Tomanek, Monika; Jastrzębska, Maria; Marciniec, Krzysztof; Chrobak, Elwira; Bębenek, Ewa; Boryczka, Stanisław |
2021 | Molecular structure, in vitro anticancer study and molecular docking of new phosphate derivatives of betulin | Chrobak, Elwira; Jastrzębska, Maria; Bębenek, Ewa; Kadela-Tomanek, Monika; Marciniec, Krzysztof; Latocha, Małgorzata; Wrzalik, Roman; Kusz, Joachim; Boryczka, Stanisław |
2017 | New acetylenic amine derivatives of 5,8-quinolinediones : synthesis, crystal structure and antiproliferative activity | Kadela-Tomanek, Monika; Jastrzębska, Maria; Bębenek, Ewa; Chrobak, Elwira; Latocha, Małgorzata; Kusz, Joachim; Tarnawska, Dorota; Boryczka, Stanisław |
2019 | New phosphorus analogs of bevirimat: synthesis, evaluation of anti-HIV-1 activity and molecular docking study | Chrobak, Elwira; Marciniec, Krzysztof; Dąbrowska, Aleksandra; Pęcak, Paweł; Bębenek, Ewa; Kadela-Tomanek, Monika; Bąk, Andrzej; Jastrzębska, Maria; Boryczka, Stanisław |
2017 | Novel triazole hybrids of betulin : synthesis and biological activity profile | Bębenek, Ewa; Jastrzębska, Maria; Kadela-Tomanek, Monika; Chrobak, Elwira; Orzechowska, Beata; Zwolińska, Katarzyna; Latocha, Małgorzata; Mertas, Anna; Czuba, Zenon; Boryczka, Stanisław |
2021 | Spectroscopic investigations, computational analysis and molecular docking to SAR-Cov-2 targets studies of 5,8-quinolinedione attached to betulin derivatives | Kadela-Tomanek, Monika; Jastrzębska, Maria; Marciniec, Krzysztof; Bębenek, Ewa; Chrobak, Elwira; Boryczka, Stanisław |
2018 | Structural determinants influencing halogen bonding : a case study on azinesulfonamide analogs of aripiprazole as 5-HT1A, 5-HT7, and D2 receptor ligands | Marciniec, Krzysztof; Kurczab, Rafał; Książek, Maria; Bębenek, Ewa; Chrobak, Elwira; Satała, Grzegorz; Bojarski, Andrzej J.; Kusz, Joachim; Zajdel, Paweł |
2022 | Synthesis and Structural Characterization of a New 1,2,3-Triazole Derivative of Pentacyclic Triterpene | Bębenek, Ewa; Kadela-Tomanek, Monika; Chrobak, Elwira; Jastrzębska, Maria; Książek, Maria |
2016 | Synthesis, structure and cytotoxic activity of mono- and dialkoxy derivatives of 5,8-quinolinedione | Kadela, Monika; Jastrzębska, Maria; Bębenek, Ewa; Chrobak, Elwira; Latocha, Małgorzata; Kusz, Joachim; Książek, Maria; Boryczka, Stanisław |
2013 | Synthesis, structure and cytotoxic activity of new acetylenic derivatives of betulin | Boryczka, Stanisław; Bębenek, Ewa; Wietrzyk, Joanna; Kempińska, Katarzyna; Jastrzębska, Maria; Kusz, Joachim; Nowak, Maria |